Signaling peptide receptor

Signaling peptide receptor is a type of receptor which binds one or more signaling peptides or signaling proteins.

An example is the tropomyosin receptor kinase B (TrkB), which is bound and activated by the neurotrophic protein brain-derived neurotrophic factor (BDNF). Another example is the μ-opioid receptor (MOR), which is bound and activated by the opioid peptide hormone β-endorphin.

Adiponectin receptor

AdipoR1

  • Agonists
    • Peptide
    • Non-peptide
      • AdipoRon
      • (–)-Arctigenin
      • Arctiin
      • Gramine
      • Matairesinol
  • Antagonists
    • Peptide
      • ADP-400

AdipoR2

  • Agonists
  • Antagonists
    • Peptide
      • ADP-400

Angiotensin receptor

Bradykinin receptor

  • Agonists
  • Antagonists
    • FR-173657
    • Icatibant
    • LF22-0542
  • Agonists
  • Antagonists
    • Atogepant
    • BI 44370 TA
    • CGRP (8-37)
    • MK-3207
    • Olcegepant
    • Rimegepant
    • SB-268262
    • Telcagepant
    • Ubrogepant
  • Antibodies
    • Eptinezumab
    • Erenumab
    • Fremanezumab
    • Galcanezumab

Cholecystokinin receptor

CCKA

  • Agonists
  • Antagonists
    • Amiglumide
    • Asperlicin
    • Devazepide
    • Dexloxiglumide
    • Lintitript
    • Lorglumide
    • Loxiglumide
    • Pranazepide
    • Proglumide
    • Tarazepide
    • Tomoglumide

CCKB

Unsorted

  • Antagonists
    • Nastorazepide

Corticotropin-releasing hormone receptor

CRF1

CRF2

Cytokine receptor

Endothelin receptor

  • Agonists
  • Antagonists
    • A-192621
    • Ambrisentan
    • Aprocitentan
    • Atrasentan
    • Avosentan
    • Bosentan
    • BQ-123
    • BQ-788
    • Clazosentan
    • Darusentan
    • Edonentan
    • Enrasentan
    • Fandosentan
    • Feloprentan
    • Macitentan
    • Nebentan
    • Sitaxentan
    • Sparsentan
    • Tezosentan
    • Zibotentan

Galanin receptor

GAL1

  • Agonists
  • Antagonists
    • C7
    • Dithiepine-1,1,4,4-tetroxide
    • Galantide (M15)
    • M32
    • M35
    • M40
    • SCH-202596

GAL2

  • Agonists
  • Antagonists
    • C7
    • Galantide (M15)
    • M32
    • M35
    • M40
    • M871

GAL3

  • Agonists
    • Galanin
    • Galanin (1-15)
    • Galmic
    • Galnon
  • Antagonists
    • C7
    • Galantide (M15)
    • GalR3ant
    • HT-2157
    • M32
    • M35
    • M40
    • SNAP-37889
    • SNAP-398299

Growth hormone secretagogue receptor

Growth hormone receptor

Growth-hormone-releasing hormone receptor

Glucagon-like peptide receptor

GLP-1

  • Agonists
    • Albiglutide
    • Beinaglutide
    • Dulaglutide
    • Efpeglenatide
    • Exenatide
    • GLP-1
    • Langlenatide
    • Liraglutide
    • Lixisenatide
    • Oxyntomodulin
    • Pegapamodutide
    • Semaglutide
    • Taspoglutide

GLP-2

  • Agonists
    • Apraglutide
    • Elsiglutide
    • Glepaglutide
    • GLP-2
    • Teduglutide

Others

Glucagon receptor

Gonadotropin-releasing hormone receptor

Gonadotropin receptor

Growth factor receptor

Insulin receptor

  • Agonists
  • Antagonists
    • BMS-754807
    • S661
    • S961
  • Kinase inhibitors
    • Linsitinib
  • Antibodies
    • Xentuzumab (against IGF-1 and IGF-2)

KiSS1-derived peptide receptor

Leptin receptor

Melanin-concentrating hormone receptor

MCH1

MCH2

Melanocortin receptor

Neuropeptide FF receptor

  • Agonists
    • Neuropeptide AF
    • Neuropeptide FF
    • Neuropeptide SF (RFRP-1)
    • Neuropeptide VF (RFRP-3)
  • Antagonists
    • BIBP-3226
    • RF9

Neuropeptide S receptor

Neuropeptide Y receptor

Y1

Y2

  • Agonists
  • Antagonists
    • BIIE-0246
    • JNJ-5207787
    • SF-11

Y4

Y5

  • Agonists
  • Antagonists
    • CGP-71683
    • FMS-586
    • L-152,804
    • Lu AA-33810
    • MK-0557
    • NTNCB
    • Velneperit (S-2367)

Neurotensin receptor

NTS1

NTS2

  • Agonists
  • Antagonists
    • Levocabastine
      • SR-142948

Opioid receptor

Orexin receptor

Oxytocin receptor

Prolactin receptor

Parathyroid hormone receptor

Relaxin receptor

Somatostatin receptor

Tachykinin receptor

Thyrotropin-releasing hormone receptor

  • Agonists
    • Azetirelin
    • JTP-2942
    • Montirelin
    • Orotirelin
    • Posatirelin
    • Protirelin
    • Rovatirelin
    • RX-77368 (thymoliberin)
    • Taltirelin
    • TRH (TRF)

Thyrotropin receptor

Vasopressin receptor

Vasoactive intestinal peptide receptor and Pituitary adenylate cyclase-activating peptide

VIPR1

  • Agonists

VIPR2

PAC1

  • Agonists
    • PACAP
    • PACAP (1-27)
    • PACAP (1-38)
  • Antagonists
    • PACAP (6-38)

Unsorted

Others

See also

References

    This article is issued from Wikipedia. The text is licensed under Creative Commons - Attribution - Sharealike. Additional terms may apply for the media files.